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Current Pharmaceutical Design

Editor-in-Chief

ISSN (Print): 1381-6128
ISSN (Online): 1873-4286

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Editorial

Progress in the Development of Agonists, Antagonists and Allosteric Modulators of Adenosine Receptors

Author(s): Pran Kishore Deb

Volume 25, Issue 25, 2019

Page: [2695 - 2696] Pages: 2

DOI: 10.2174/138161282525190916100149

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Chandrasekaran B, Deb PK, Kachler S, Akkinepalli RR, Mailavaram R, Klotz K-N. Synthesis and adenosine receptors binding studies of new fluorinated analogues of pyrido [2,3-d]pyrimidines and quinazolines. Med Chem Res 2018; 27: 756-67.
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Deb PK. Recent Updates in the Computer Aided Drug Design Strategies for the Discovery of Agonists and Antagonists of Adenosine Receptors. In: ed. Bentham Science 2019; 747-9.
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Deb PK, Chandrasekaran B, Mailavaram R, Tekade RK, Jaber AMY. Molecular modeling approaches for the discovery of adenosine A2B receptor antagonists: current status and future perspectives. Drug Discov Today 2019; pii: S1359-6446(19): 30045-5.
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Deb PK, Balakumar C, Rao AR, Roy PP, Roy K. QSAR of adenosine receptor antagonists: exploring physicochemical requirements for binding of pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives with human adenosine A3 receptor subtype. Bioorg Med Chem Lett 2011; 21: 818-23.
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Deb PK, Deka S, Borah P, Abed SN, Klotz K-N. Medicinal chemistry and therapeutic potential of agonists, antagonists and allosteric modulators of A1 adenosine receptor: current status and perspectives. Curr Pharm Des 2019; 25(25): 2697-715.
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Chandrasekaran B, Samarneh S, Kassab G, Agrawal N. Therapeutic potentials of A2B adenosine receptor ligands: Current status and perspectives. Curr Pharm Des 2019; 25(25): 2741-71.
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Mailavaram RP, Al-Attraqchi OHA, Kar S, Ghosh S. Current status in the design and development of agonists and antagonists of adenosine A3 receptor as potential therapeutic agents. Curr Pharm Des 2019; 25(25): 2772-87.

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