Search Result "Aminobutyric acid(A) receptors"


Research Article

Microwave Assisted Synthesis and Molecular Docking Studies of Some 4 - (3H)-quinazolinone Derivatives as Inhibitors of Human Gamma- Aminobutyric Acid Receptor, the GABA (A)R-BETA3 Homopentamer

Journal: Medicinal Chemistry
Volume: 17 Issue: 5 Year: 2021 Page: 453-461
Author(s): Amrutkar Rakesh Devidas,Mahendra Sing Ranawat

An Updated Unified Pharmacophore Model of the Benzodiazepine Binding Site on γ-Aminobutyric Acida Receptors: Correlation with Comparative Models

Journal: Current Medicinal Chemistry
Volume: 14 Issue: 2 Year: 2007 Page: 2755-2775
Author(s): T. Clayton, J. L. Chen, M. Ernst, L. Richter, B. A. Cromer, C. J. Morton, H. Ng, C. C. Kaczorowski, F. J. Helmstetter, R. Furtmuller, G. Ecker, M. W. Parker, W. Sieghart, J. M. Cook

The Four Human γ-Aminobutyric Acid (GABA) Transporters: Pharmacological Characterization and Validation of a Highly Efficient Screening Assay

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 12 Issue: 3 Year: 2009 Page: 241-249
Author(s): Trine Kvist, Bolette Christiansen, Anders A. Jensen, Hans Brauner-Osborne

Selected PET Radioligands for Ion Channel Linked Neuroreceptor Imaging: Focus on GABA, NMDA and nACh Receptors

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 16 Year: 2016 Page: 1830-1842
Author(s): Alina Kassenbrock,Neil Vasdev,Steven H. Liang

GABAB Receptors as Potential Therapeutic Targets

Journal: Current Drug Targets - CNS & Neurological Disorders
Volume: 2 Issue: 4 Year: 2003 Page: 248-259
Author(s): Claire-Marie Vacher, Bernhard Bettler

Structure, Pharmacology and Therapeutic Prospects of Family C G-Protein Coupled Receptors

Journal: Current Drug Targets
Volume: 8 Issue: 1 Year: 2007 Page: 169-184
Author(s): Hans Brauner-Osborne, Petrine Wellendorph, Anders A. Jensen

Research Article

Brain Targeted Intranasal Zaleplon Nano-emulsion: In-Vitro Characterization and Assessment of Gamma Aminobutyric Acid Levels in Rabbits’ Brain and Plasma at Low and High Doses

Journal: Current Drug Delivery
Volume: 15 Issue: 6 Year: 2018 Page: 898-906
Author(s): Eman Abd-Elrasheed,Sara Nageeb El-Helaly,Manal M. EL-Ashmoony,Salwa Salah

Derivatives of 1,2,3,4-tetrahydroisoquinoline-7-carboxylic Acid as Novel Fibrinogen Receptor Antagonists

Journal: Medicinal Chemistry
Volume: 5 Issue: 2 Year: 2009 Page: 158-164
Author(s): Olga L. Malovichko, Andrei A. Krysko, Tatyana A. Kabanova, Sergei A. Andronati, Vladimir I. Grishkovets, Vadim V. Kachala, Denis A. Panov

Assessing Structure, Function and Druggability of Major Inhibitory Neurotransmitter γ-Aminobutyrate Symporter Subtypes

Journal: Current Medicinal Chemistry
Volume: 17 Issue: 2 Year: 2010 Page: 2203-2213
Author(s): J. Kardos, A. Pallo, A. Bencsura, A. Simon

The Benzodiazepine Recognition Site on GABAA Receptors

Journal: Medicinal Chemistry Reviews - Online (Discontinued)
Volume: 2 Issue: 3 Year: 2005 Page: 251-256
Author(s): Erwin Sigel

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