Search Result "2H and 3H Labeling"


New Anticonvulsant Agents

Journal: Current Topics in Medicinal Chemistry
Volume: 5 Issue: 1 Year: 2005 Page: 69-85
Author(s): Barbara Malawska

Synthesis of 12-Deuterated and Tritiated Deoxoartemisinins

Journal: Medicinal Chemistry
Volume: 1 Issue: 2 Year: 2005 Page: 105-107
Author(s): Mankil Jung, Kyunghoon Lee

A Novel Achiral seco-Amino-Cyclopropylindoline (CI) Analog of CC-1065 and the Duocarmycins: Design, Synthesis and Biological Studies

Journal: Medicinal Chemistry
Volume: 1 Issue: 1 Year: 2005 Page: 13-19
Author(s): James L. Toth, John D. Trzupek, Lloyd V. Flores, Konstantinos Kiakos, John A. Hartley, William T. Pennington, Moses Lee

Variously Substituted (Phosphonoacetamido)Oxy Analogues of Geranylgeranyl Diphosphate (GGdP) as GGdP-transferase (GGTase) Inhibitors and Antiproliferative Agents

Journal: Medicinal Chemistry
Volume: 1 Issue: 3 Year: 2005 Page: 239-244
Author(s): Filippo Minutolo, Valentina Asso, Simone Bertini, Laura Betti, Massimiliano Ciriaco, Romano Danesi, Gianbattista Gervasi, Elisa Ghilardi, Elisa Giovanetti, Gino Giannaccini

Influence of Trishomocubanes on Sigma Receptor Binding of N-(1-Benzylpiperidin- 4-yl)-4-[123I]iodobenzamide In Vivo in the Rat Brain

Journal: Medicinal Chemistry
Volume: 1 Issue: 1 Year: 2005 Page: 31-38
Author(s): Xiang Liu, Filomena Mattner, Andrew Katsifis, MacDonald Christie, Michael Kassiou

N-Terminal Anthranoyl-Phenylalanine Derivatives as CCK1 Receptor Antagonists: The Final Approach

Journal: Medicinal Chemistry
Volume: 1 Issue: 5 Year: 2005 Page: 501-517
Author(s): A. Varnavas, L. Lassiani, V. Valenta, A. Ciogli, F. Gasparrini, L. Mennuni, F. Makovec

The Molecular Basis for the Mode of Action of Bicyclomycin

Journal: Current Drug Targets - Infectious Disorders
Volume: 5 Issue: 3 Year: 2005 Page: 273-295
Author(s): Harold Kohn, William Widger

8-(Heteroaryl)phenalkyl-1-Phenyl-1,3,8-triazaspiro[4.5]decan-4-ones as Opioid Receptor Modulators

Journal: Medicinal Chemistry
Volume: 1 Issue: 6 Year: 2005 Page: 601-610
Author(s): A. D. Jordan, M. J. Orsini, S. A. Middleton, P. J. Connolly, D. E. Brenneman, K. Pan, A. B. Reitz

Chemo-Enzymatic Synthesis of a Trisaccharide-Linked Peptide Aimed at Improved Drug-Delivery

Journal: Current Drug Delivery
Volume: 2 Issue: 3 Year: 2005 Page: 215-222
Author(s): Ken D. Johnstone, Manuela Dieckelmann, Michael P. Jennings, Istvan Toth, Joanne T. Blanchfield

Aminopyrimidinimino Isatin Analogues: Design and Synthesis of Novel Non- Nucleoside HIV-1 Reverse Transcriptase Inhibitors with Broad- Spectrum Anti-Microbial Properties

Journal: Medicinal Chemistry
Volume: 1 Issue: 3 Year: 2005 Page: 277-285
Author(s): Dharmarajan Sriram, Tanushree Ratan Bal, Perumal Yogeeswari

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