Search Result "Antimycobacterial properties"


Research Article

4-Hydroxy-2-pyridone Derivatives and the δ-pyrone Isostere as Novel Agents Against Mycobacterium smegmatis Biofilm Inhibitors

Journal: Medicinal Chemistry
Volume: 15 Issue: 1 Year: 2019 Page: 28-37
Author(s): Maheshkumar R. Borkar,Santosh Nandan,M N Harish Kumar,Jayashree Puttur,M Jisha,Dipankar Chatterji,Evans C. Coutinho

Research Article

Imidazole and 1,2,4-Triazole-based Derivatives Gifted with Antitubercular Activity: Cytotoxicity and Computational Assessment

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 8 Year: 2019 Page: 620-632
Author(s): Daniele Zampieri,Francesca Cateni,Mariarosa Moneghini,Marina Zacchigna,Erik Laurini,Domenico Marson,Alessandro De Logu,Adriana Sanna,Maria G. Mamolo

Research Article

Activity of N-Phenylpiperazine Derivatives Against Bacterial and Fungal Pathogens

Journal: Current Protein & Peptide Science
Volume: 20 Issue: 1 Year: 2019 Page: 1119-1129
Author(s): Sarka Pospisilova,Pavlina Marvanova,Jakub Treml,Agnes M. Moricz,Peter G. Ott,Petr Mokry,Klara Odehnalova,Ondrej Sedo,Alois Cizek,Josef Jampilek

Review Article

Recent Advances in the Chemistry and Synthesis of Thienopyrazine, Pyrrolopyrazine and Furopyrazine Derivatives

Journal: Current Organic Chemistry
Volume: 23 Issue: 2 Year: 2019 Page: 2635-2663
Author(s): Majid M. Heravi,Afsaneh Feiz,Ayoob Bazgir

Review Article

4H-1,3-Benzothiazin-4-one a Promising Class Against MDR/XDR-TB

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 8 Year: 2019 Page: 567-578
Author(s): Marcus Vinicius Nora de Souza,Thais Cristina Mendonça Nogueira

Research Article

Tryptanthrin Analogues as Inhibitors of Enoyl-acyl Carrier Protein Reductase: Activity against Mycobacterium tuberculosis, Toxicity, Modeling of Enzyme Binding

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 8 Year: 2019 Page: 609-619
Author(s): Gheorghe Duca,Serghei Pogrebnoi,Veaceslav Boldescu,Fatma Aksakal,Andrei Uncu,Vladimir Valica,Livia Uncu,Simona Negres,Florica Nicolescu,Fliur Macaev

Research Article

Design, Synthesis, Crystal Structure, Fluorescence, Molecular Docking and DFT Studies of 3,6-Dinitro-N-octylcarbazole

Journal: Current Organic Chemistry
Volume: 23 Issue: 1 Year: 2019 Page: 1681-1687
Author(s): Hummera Rafique,Aamer Saeed,Fouzia Perveen,Naghmana Kausar,Zaman Ashraf,Sadia Akram,Muhammad Naveed Zafar,Muhammad Tayyab,Ulrich Flörke

Review Article

An Overview of Recent Advances in Biological and Pharmaceutical Developments of Fluoro-containing Drugs

Journal: Current Organic Chemistry
Volume: 23 Issue: 26 Year: 2019 Page: 2916-2944
Author(s): Nader G. Khaligh,Hanna Abbo,Salam J.J. Titinchi,Mohd R. Johan

Research Article

Preparation and Antitubercular Activities of Palindromic Hydrazinecarbothioamides and Carbonothioic Dihydrazides

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 1 Year: 2019 Page: 1202-1210
Author(s): Michael Joseps Hearn,Gwendolyn Towers,Michael Henry Cynamon

Research Article

Ultrasonically Assisted Efficient and Green Protocol for the Synthesis of 4H-isoxazol-5-ones using Itaconic Acid as a Homogeneous and Reusable Organocatalyst

Journal: Current Organocatalysis
Volume: 6 Issue: 3 Year: 2019 Page: 231-237
Author(s): Sandeep B. Kasar,Shankar R. Thopate

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