Search Result "BCR-ABL"


Review Article

Unleashing the Guardian: The Targetable BCR-ABL/HAUSP/PML/PTEN Network in Chronic Myeloid Leukemia

Journal: Current Drug Targets
Volume: 18 Issue: 4 Year: 2017 Page: 389-395
Author(s): Alessandro Morotti,Davide Torti,Giovanna Carra,Cristina Panuzzo,Sabrina Crivellaro,Riccardo Taulli,Carmen Fava,Angelo Guerrasio,Giuseppe Saglio

Review Article

Development of a Predictive Pharmacophore Model and a 3D-QSAR Study for an in silico Screening of New Potent Bcr-Abl Kinase Inhibitors

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2017 Page: 188-204
Author(s): Eleni Vrontaki,Georgia Melagraki,Stella Voskou,Marios S. Phylactides,Thomas Mavromoustakos,Marina Kleanthous,Antreas Afantitis

Review Article

A Virtual Screening Approach for the Identification of High Affinity Small Molecules Targeting BCR-ABL1 Inhibitors for the Treatment of Chronic Myeloid Leukemia

Journal: Current Topics in Medicinal Chemistry
Volume: 17 Issue: 26 Year: 2017 Page: 2989-2996
Author(s): Saphy Sharda,Palash Sarmandal,Shirisha Cherukommu,Kiran Dindhoria,Manisha Yadav,Srinivas Bandaru,Anudeep Sharma,Aditi Sakhi,Tanmay Vyas,Tajamul Hussain,Anuraj Nayarisseri,Sanjeev Kumar Singh

Research Article

In Vitro Sensitivity Profiling of Neuroblastoma Cells Against A Comprehensive Small Molecule Kinase Inhibitor Library to Identify Agents for Future Therapeutic Studies

Journal: Current Cancer Drug Targets
Volume: 17 Issue: 6 Year: 2017 Page: 569-584
Author(s): Anjali Singh,Vanessa Meier-Stephenson,Aarthi Jayanthan,Aru Narendran

Review Article

Stem Cell Guardians – Old and New Perspectives in LSC Biology

Journal: Current Drug Targets
Volume: 18 Issue: 4 Year: 2017 Page: 405-413
Author(s): Gillian A. Horne,Lorna Jackson,Vignir Helgason,Tessa L. Holyoake

Research Article

Design, Synthesis and Biological Evaluation of Betulinic Acid Derivatives as New Antitumor Agents for Leukemia

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 1 Year: 2017 Page: 1777-1785
Author(s): Fernanda Waechter,Gloria N.S. da Silva,Julia B. Willig,Cristiane B. de Oliveira,Bruna D. Vieira,Daniela B.B. Trivella,Aline R. Zimmer,Andreia Buffon,Diogo A. Pilger,Simone C.B. Gnoatto

Review Article

Is Going for Cure in CML Targeting Aberrant Glycogen Synthase Kinase 3β?

Journal: Current Drug Targets
Volume: 18 Issue: 4 Year: 2017 Page: 396-404
Author(s): Concetta Saponaro,Michele Maffia,Nicola Di Renzo,Addolorata Maria Luce Coluccia

Review Article

The Polyhedric Abl Kinases and their Pharmacologic Inhibitors

Journal: Current Enzyme Inhibition
Volume: 13 Issue: 2 Year: 2017 Page: 129-138
Author(s): Elisa Lupino, Marco Piccinini

Review Article

Multi-Targeted Anticancer Agents

Journal: Current Topics in Medicinal Chemistry
Volume: 17 Issue: 28 Year: 2017 Page: 3084-3098
Author(s): Wei Zheng,Yao Zhao,Qun Luo,Yang Zhang,Kui Wu,Fuyi Wang

Editorial free to download

Editorial (Thematic Issue: CML HSCs: Are the True Enemies for the Patient?)

Journal: Current Drug Targets
Volume: 18 Issue: 4 Year: 2017 Page: 376-376
Author(s): Manuela Mancini

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