Search Result "HDAC"


Review Article

Histone Deacetylases (HDACs) in Gastric Cancer: An Update of Their Emerging Prognostic and Therapeutic Role

Journal: Current Medicinal Chemistry
Volume: 27 Issue: 3 Year: 2020 Page: 6099-6111
Author(s): Dimitrios Schizas,Aikaterini Mastoraki,Leon Naar,Diamantis I. Tsilimigras,Ioannis Katsaros,Vasiliki Fragkiadaki,Georgia-Sofia Karachaliou,Nikolaos Arkadopoulos,Theodore Liakakos,Dimitrios Moris

Review Article

Recent Studies on HDAC Inhibitors Acting against Prostate Cancer

Journal: Current Enzyme Inhibition
Volume: 16 Issue: 1 Year: 2020 Page: 74-89
Author(s): Basheerulla Shaik,Tabassum Zafar,Satya P. Gupta

Review Article

Epidermal Growth Factor Receptor and its Trafficking Regulation by Acetylation: Implication in Resistance and Exploring the Newer Therapeutic Avenues in Cancer

Journal: Current Topics in Medicinal Chemistry
Volume: 20 Issue: 1 Year: 2020 Page: 1105-1123
Author(s): Manvendra Kumar,Gaurav Joshi,Joydeep Chatterjee,Raj Kumar

Review Article

Recent Progress in Histone Deacetylase Inhibitors as Anticancer Agents

Journal: Current Medicinal Chemistry
Volume: 27 Issue: 1 Year: 2020 Page: 2449-2493
Author(s): Loredana Cappellacci,Diego R. Perinelli,Filippo Maggi,Mario Grifantini,Riccardo Petrelli

Research Article

Searching for Potential HDAC2 Inhibitors: Structure-activity Relationship Studies on Indole-based Hydroxamic Acids as an Anticancer Agent

Journal: Letters in Drug Design & Discovery
Volume: 17 Issue: 7 Year: 2020 Page: 905-917
Author(s): Ekta Shirbhate,Divya,Preeti Patel,Vijay K. Patel,Ravichandran Veerasamy,Prabodh C. Sharma,Harish Rajak

Research Article

Synthesis and Evaluation of 18F-INER-1577-3 as a Central Nervous System (CNS) Histone Deacetylase Imaging Agent

Journal: Current Medical Imaging
Volume: 16 Issue: 8 Year: 2020 Page: 978-990
Author(s): Ming-Hsin Li,Han-Chih Chang,Chun-Fang Feng,Hung-Wen Yu,Chyng-Yann Shiue

Research Article

Epigenetic Evaluation of N-(2-hydroxyphenyl)-2-Propylpentanamide, a Valproic Acid Aryl Derivative with Activity Against HeLa Cells

Journal: Current Molecular Pharmacology
Volume: 13 Issue: 0 Year: 2020 Page: 1-9
Author(s): Luna-Palencia Gabriela Rebeca,Correa-Basurto José,Trujillo-Ferrara José,Meraz-Ríos Marco Antonio,Vásquez-Moctezuma Ismael

Review Article

Novel Selective Histone Deacetylase 6 (HDAC6) Inhibitors: A Patent Review (2016-2019)

Journal: Recent Patents on Anti-Cancer Drug Discovery
Volume: 15 Issue: 1 Year: 2020 Page: 32-48
Author(s): Xingrui He,Zhen Li,Xiao-Tao Zhuo,Zi Hui,Tian Xie,Xiang-Yang Ye

Research Article

Histone Deacetylase Inhibitor Trichostatin A Suppresses Cell Proliferation and Induces Apoptosis by Regulating the PI3K/AKT Signalling Pathway in Gastric Cancer Cells

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 20 Issue: 1 Year: 2020 Page: 2114-2124
Author(s): Xinli An,Zekun Wei,Botian Ran,Hao Tian,Hongyu Gu,Yan Liu,Hongjuan Cui,Shunqin Zhu

General Research Article

Cinnamyl Sulfonamide Hydroxamate Derivatives Inhibited LPS-Stimulated NF-kB Expression in RAW 264.7 Cells In Vitro and Mitigated Experimental Colitis in Wistar Rats In Vivo

Journal: Current Pharmaceutical Design
Volume: 26 Issue: 3 Year: 2020 Page: 4934-4943
Author(s): Mit Joshi,Neetinkumar D. Reddy,Nitesh Kumar,Suhani Sumalatha,C. Mallikarjuna Rao

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