Search Result "MDR"


Promising Therapy of XDR-TB/MDR-TB with Thioridazine an Inhibitor of Bacterial Efflux Pumps

Journal: Current Drug Targets
Volume: 9 Issue: 9 Year: 2008 Page: 816-819
Author(s): L. Amaral, M. Martins, M. Viveiros, J. Molnar, J. E. Kristiansen

Synthesis of 2-Methyl N10-Substituted Acridones as Selective Inhibitors of Multidrug Resistance (MDR) Associated Protein in Cancer Cells

Journal: Medicinal Chemistry
Volume: 4 Issue: 5 Year: 2008 Page: 457-465
Author(s): Y. C. Mayur, Osman Ahmad, V. V.S. Rajendra Prasad, M. N. Purohit, N. Srinivasulu, S. M. Shanta Kumar

New Methods for the Identification of Efflux Mediated MDR Bacteria, Genetic Assessment of Regulators and Efflux Pump Constituents, Characterization of Efflux Systems and Screening for Inhibitors of Efflux Pumps

Journal: Current Drug Targets
Volume: 9 Issue: 9 Year: 2008 Page: 760-778
Author(s): M. Viveiros, M. Martins, I. Couto, L. Rodrigues, G. Spengler, A. Martins, J. E. Kristiansen, J. Molnar, L. Amaral

Strategies to Overcome or Circumvent P-Glycoprotein Mediated Multidrug Resistance

Journal: Current Medicinal Chemistry
Volume: 15 Issue: 5 Year: 2008 Page: 470-476
Author(s): Xun Li, Hongyu Yuan, Jifeng Wu, Jinpei Li, Xianjun Qu, Wenfang Xu, Wei Tang

Clinical Impact of the Over-Expression of Efflux Pump in Nonfermentative Gram-Negative Bacilli, Development of Efflux Pump Inhibitors

Journal: Current Drug Targets
Volume: 9 Issue: 9 Year: 2008 Page: 797-807
Author(s): Jordi Vila, Jose Luis Martinez

Anti-Mycobacterial Activity of Quinolones. Triazoloquinolones a New Class of Potent Anti-Mycobacterial Agents

Journal: Anti-Infective Agents in Medicinal Chemistry
Volume: 7 Issue: 2 Year: 2008 Page: 134-147
Author(s): Antonio Carta, Sandra Piras, Michele Palomba, Daniela Jabes, Paola Molicotti, Stefania Zanetti

Editorial [Hot topic: Control and Regulation of Permeability of MDR Bacterial Pathogens to Antibiotics Presented by COST Action BM0701 (Guest Editors: L. Amaral and J.M. Pages)]

Journal: Current Drug Targets
Volume: 9 Issue: 9 Year: 2008 Page: 718-718
Author(s): Leonard Amaral, Jean Marie Pages

Synthesis, Antimycobacterial Activities and Phototoxic Evaluation of 5H-thiazolo[3,2-a]quinoline-4-carboxylic Acid Derivatives

Journal: Medicinal Chemistry
Volume: 4 Issue: 5 Year: 2008 Page: 482-491
Author(s): Murugesan Dinakaran, Palaniappan Senthilkumar, Perumal Yogeeswari, Arnab China, Valakunja Nagaraja, Dharmarajan Sriram

Membrane Permeability and Regulation of Drug “Influx and Efflux” in Enterobacterial Pathogens

Journal: Current Drug Targets
Volume: 9 Issue: 9 Year: 2008 Page: 750-759
Author(s): Anne Davin-Regli, Jean-Michel Bolla, Chloe E. James, Jean-Philippe Lavigne, Jacqueline Chevalier, Eric Garnotel, Alexander Molitor, Jean-Marie Pages

Reversal of ABC Drug Transporter-Mediated Multidrug Resistance in Cancer Cells: Evaluation of Current Strategies

Journal: Current Molecular Pharmacology
Volume: 1 Issue: 2 Year: 2008 Page: 93-105
Author(s): Chung-Pu Wu, Anna Maria Calcagno, Suresh V. Ambudkar

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