Search Result "P-glycoprotein efflux transport"


Research Article

Exploring the Chemical Space of P-Glycoprotein Interacting Compounds

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 17 Issue: 14 Year: 2017 Page: 1332-1345
Author(s): Veda Prachayasittikul,Prasit Mandi,Supaluk Prachayasittikul,Virapong Prachayasittikul,Chanin Nantasenamat

Review Article

Phenothiazines and Related Drugs as Multi Drug Resistance Reversal Agents in Cancer Chemotherapy Mediated by p-glycoprotein

Journal: Current Cancer Therapy Reviews
Volume: 13 Issue: 1 Year: 2017 Page: 28-42
Author(s): Ravinesh Mishra,Swati Sareen,Bhartendu Sharma,Shubham Goyal,Gurpreet Kaur,Sweta Bhardwaj,Anees A. Siddiqui,Asif Husain,Rajeev K. Singla,Mohd Rashid,Deepak Kumar,Bhawana Sati,Nishtha Shalmali,Rajiv Kumar

Research Article

Quantitative Structure Activity Relationship (QSAR) of Methylated Polyphenol Derivatives as Permeability Glycoprotein (P-gp) Inhibitors: A Comparison of Different Training and Test Set Selection Methods

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 9 Year: 2017 Page: 999-1007
Author(s): Paria Ghaemian,Ali Shayanfar

Review Article

Computer-Aided Recognition of ABC Transporters Substrates and Its Application to the Development of New Drugs for Refractory Epilepsy

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2017 Page: 205-215
Author(s): Manuel Couyoupetrou,Melisa E. Gantner,Mauricio E. Di Ianni,Pablo H. Palestro,Andrea V. Enrique,Luciana Gavernet,Maria E. Ruiz,Guido Pesce,Luis E. Bruno-Blanch,Alan Talevi

Review Article

Opioids and the Blood-Brain Barrier: A Dynamic Interaction with Consequences on Drug Disposition in Brain

Journal: Current Neuropharmacology
Volume: 15 Issue: 8 Year: 2017 Page: 1156-1173
Author(s): Catarina Chaves,Fernando Remiao,Salvatore Cisternino,Xavier Decleves

Research Article

Grid-independent Descriptors (GRIND) Analysis and SAR Guided Molecular Docking Studies to Probe Selectivity Profiles of Inhibitors of Multidrug Resistance Transporters ABCB1 and ABCG2

Journal: Current Cancer Drug Targets
Volume: 17 Issue: 2 Year: 2017 Page: 177-190
Author(s): Talha Shafi,Ishrat Jabeen

Review Article

The Role of Metabolizing Enzymes and Transporters in Antiretroviral Therapy

Journal: Current Topics in Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2017 Page: 340-360
Author(s): Ling Ye,Chuqi Hou,Shuwen Liu

Drug Delivery to the Brain by Liposomal Carrier Systems

Ebook: Frontiers in Nanomedicine

Volume: 2 Year: 2017
Author(s): Anne Mahringer,Gert Fricker
Doi: 10.2174/9781681084930117020007
Review Article

MRP1-dependent Collateral Sensitivity of Multidrug-resistant Cancer Cells: Identifying Selective Modulators Inducing Cellular Glutathione Depletion

Journal: Current Medicinal Chemistry
Volume: 24 Issue: 1 Year: 2017 Page: 1186-1213
Author(s): Doriane Lorendeau,Lauriane Dury,Rachad Nasr,Ahcene Boumendjel,Elisabetta Teodori,Michael Gutschow,Pierre Falson,Attilio Di Pietro,Helene Baubichon-Cortay

Review Article

Nanomedicine to Deal With Cancer Cell Biology in Multi-Drug Resistance

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 17 Issue: 18 Year: 2017 Page: 1793-1810
Author(s): Pawan Tekchandani,Balak Das Kurmi,Shivani Rai Paliwal

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