Search Result "Quinazolinone"


Review Article

Antileishmanial Drug Discovery: Synthetic Methods, Chemical Characteristics, and Biological Potential of Quinazolines and its Derivatives

Journal: Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry
Volume: 16 Issue: 1 Year: 2017 Page: 3-32
Author(s): Adarsh Sahu,Deepak Kumar,Ram Kishore Agrawal

Research Article

Synthesis and Evaluation of Some Dibromoquinazoline-sulphonamide Hybrids and some Schiff´s Base Analogs for their Cytotoxic Activity

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 11 Year: 2017 Page: 1563-1569
Author(s): Marwa F. Ahmed,Radwan El-Haggar

Research Article

Alkaline Starch as a New Biocompatible Base Catalyst for Improved Multi-Strategic Synthesis of Hydroquinazolinones

Journal: Current Catalysis
Volume: 6 Issue: 1 Year: 2017 Page: 57-66
Author(s): Fatemeh Tamaddon, Mohammad Taghi Kazemi Varnamkhasti

Research Article

Design and Synthesis of 4-substituted Quinazolines as Potent EGFR Inhibitors with Anti-breast Cancer Activity

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 6 Year: 2017 Page: 832-838
Author(s): Marwa F. Ahmed,Naja Magdy

Review Article

Isocyanide-based Cascade Reactions in the Synthesis of Aza-heterocycles: A Marriage of Convenience

Journal: Current Organic Chemistry
Volume: 21 Issue: 15 Year: 2017 Page: 1440-1529
Author(s): Majid M. Heravi,Niousha Nazari

Research Article

Development of Novel Selective Pharmacophore for Tankyrase Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 10 Year: 2017 Page: 1164-1175
Author(s): Xin Qiao,Ting Ran,Yan-Min Zhang,Jing Pan,Ling-Feng Yin,Wei-Neng Zhou,Lu Zhu,Jun-Nan Zhao,Hai-Chun Liu,Shuai Lu,Tao Lu,Ya-Dong Chen,Yu-Lei Jiang

Research Article

Bisthiourea Derivatives of Dipeptide Conjugated Benzo[d]isoxazole as a New Class of Therapeutics: Synthesis and Molecular Docking Studies

Journal: Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2017 Page: 123-133
Author(s): Honnegowdanahally K. Kumara,Doddahindaiah M. Suyoga Vardhan,J. Shiva Kumar,D. Channe Gowda

Research Article

Polymer-supported (-)-8-phenylmenthyl Auxiliary as an Effective Solidphase Chiral Inductor in the Addition of Nucleophiles to N-acyliminium Ions

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 20 Issue: 8 Year: 2017 Page: 696-702
Author(s): Oscar Forero-Doria,Leonardo S. Santos,Fabiane M. Nachtigall,Nagula Shankaraiah

Review Article

PDE7-Selective and Dual Inhibitors: Advances in Chemical and Biological Research

Journal: Current Medicinal Chemistry
Volume: 24 Issue: 7 Year: 2017 Page: 673-700
Author(s): Agnieszka Jankowska,Artur Swierczek,Grazyna Chlon-Rzepa,Maciej Pawlowski,Elzbieta Wyska

Review Article

Phosphoinositide-3-kinases as the Novel Therapeutic Targets for the Inflammatory Diseases: Current and Future Perspectives

Journal: Current Drug Targets
Volume: 18 Issue: 14 Year: 2017 Page: 1622-1640
Author(s): Preeti Vyas,Divya Vohora

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