Search Result "bioisosterism"


Benzenecarboxamide Analogs of Fluoroquinolones (BCFQs). Antibacterial Activity and SAR Studies

Journal: Letters in Drug Design & Discovery
Volume: 3 Issue: 2 Year: 2006 Page: 108-111
Author(s): M. J. Nieto, F. L. Alovero, R. H. Manzo, M. R. Mazzieri

Targeting Calmodulin in Reversing Multi Drug Resistance in Cancer Cells

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 6 Issue: 1 Year: 2006 Page: 1383-1389
Author(s): Y. C. Mayur, S. Jagadeesh, K. N. Thimmaiah

Medicinal Chemistry of N-Acylhydrazones: New Lead-Compounds of Analgesic, Antiinflammatory and Antithrombotic Drugs

Journal: Current Medicinal Chemistry
Volume: 13 Issue: 2 Year: 2006 Page: 167-198
Author(s): Carlos A.M. Fraga, Eliezer J. Barreiro

Editorial [ Hot Topics in Diazine Chemistry (Guest Editor: Peter Matyus)]

Journal: Current Organic Chemistry
Volume: 10 Issue: 3 Year: 2006 Page: 257-257
Author(s): Peter Matyus

Novel Fibrinogen Receptor Antagonists - RGDF Mimetics, 4-(1,2,3,4- tetrahydro-isoquinoline-7-yl)amino-4-oxo-butyric Acid Derivatives

Journal: Medicinal Chemistry
Volume: 2 Issue: 3 Year: 2006 Page: 295-298
Author(s): Sergei A. Andronati, Olga L. Malovichko, Andrei A. Krysko, Tatyana A. Kabanova, Tamara L. Karaseva, Anna S. Petrus

Silicon Switches of Marketed Drugs

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 6 Issue: 1 Year: 2006 Page: 1169-1177
Author(s): P. K. Pooni, G. A. Showell

Initial Design and Synthesis of Conformationally Restricted and Pharmacophore-Based Scaffold Hopping Analogs of a Ras Pathway Modulator and Evaluation of Their MAPK Inhibitory Activities

Journal: Letters in Drug Design & Discovery
Volume: 3 Issue: 1 Year: 2006 Page: 44-48
Author(s): Sukumar Sakamuri, Quin-Zene Chen, Yingchun Lu, Yen-Fang Keng, Vladimir Khazak, Katrin Illgen, Silke Schabbert, Lutz Weber, Sanjay R. Menon

Practical Outcome of Azaphthalimide Reduction with Zn/AcOH at Various Temperatures

Journal: Letters in Organic Chemistry
Volume: 3 Issue: 5 Year: 2006 Page: 379-383
Author(s): Mikhail Krasavin, Dmitry V. Kravchenko, Tatiana D. Talismanova, Vladimir V. Koleda, Olga Ushakova, Vladislav Z. Parchinsky

Structure-Activity Relationships of Selective GABA Uptake Inhibitors

Journal: Current Topics in Medicinal Chemistry
Volume: 6 Issue: 1 Year: 2006 Page: 1861-1882
Author(s): Signe Hog, Jeremy R. Greenwood, Karsten B. Madsen, Orla M. Larsson, Bente Frolund, Arne Schousboe, Povl Krogsgaard-Larsen, Rasmus P. Clausen

In vitro Anti-Mycobacterial Activities of Various 2-Deoxyuridine, 2- Arabinouridine and 2-Arabinofluoro-2-deoxyuridine Analogues: Synthesis and Biological Studies

Journal: Medicinal Chemistry
Volume: 2 Issue: 3 Year: 2006 Page: 287-293
Author(s): Rakesh Kumar, Dennis Y. Kunimoto, Tracey Manning, Naveen C. Srivastav

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