Search Result "checkpoint inhibition"


Kinase CK2 Inhibition: An Update

Journal: Current Medicinal Chemistry
Volume: 20 Issue: 5 Year: 2013 Page: 671-693
Author(s): G. Cozza, L. A. Pinna, S. Moro

Inhibition of Akt/mTOR Signaling by the Dietary Flavonoid Fisetin

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 13 Issue: 7 Year: 2013 Page: 995-1001
Author(s): Deeba N. Syed, Vaqar M. Adhami, Mohammad Imran Khan, Hasan Mukhtar

Targeting the Ubiquitin Proteasome System: Beyond Proteasome Inhibition

Journal: Current Pharmaceutical Design
Volume: 19 Issue: 2 Year: 2013 Page: 4053-4093
Author(s):

Protein Kinase C Modulates Aurora-kinase Inhibition Induced by CCT129202 in HMC-1560,816 Cell Line

Journal: Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry
Volume: 12 Issue: 3 Year: 2013 Page: 265-276
Author(s): Araceli Tobio, Amparo Alfonso, Andrea Fernandez-Araujo, Eva Alonso, Luis M. Botana

Dual Inhibition of PI3-Kinase and mTOR in Renal Cell Carcinoma

Journal: Current Cancer Drug Targets
Volume: 13 Issue: 2 Year: 2013 Page: 126-142
Author(s): Daniel C. Cho, James W. Mier

Antitumoral Activity of Indole-3-carbinol Cyclic tri- and Tetrameric Derivatives Mixture in Human Breast Cancer Cells: In Vitro and In Vivo Studies

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 13 Issue: 4 Year: 2013 Page: 654-662
Author(s): Giorgio Brandi, Alessandra Fraternale, Simone Lucarini, Mirko Paiardini, Mauro De Santi, Barbara Cervasi, Maria F. Paoletti, Luca Galluzzi, Andrea Duranti, Mauro Magnani

The Therapeutical Potential of a Novel Pterocarpanquinone LQB-118 to Target Inhibitor of Apoptosis Proteins in Acute Myeloid Leukemia Cells

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 13 Issue: 2 Year: 2013 Page: 341-351
Author(s): Flaviana R. de Souza Reis,Fernanda C. Casal de Faria,Carolina P. Castro,Paloma S. de Souza,Flavia da Cunha Vasconcelos,Reinaldo D. Bello,Alcides J. da Silva,Paulo R.R. Costa,Raquel C. Maia

Modulation of Arachidonic Acid Metabolism in Niemann-Pick Disease Type C Cells

Journal: Current Psychopharmacology
Volume: 2 Issue: 1 Year: 2013 Page: 58-65
Author(s): Hiroyuki Nakamura

Synthesis, p38 Kinase Inhibitory and Anti-inflammatory Activity of New Substituted Benzimidazole Derivatives

Journal: Medicinal Chemistry
Volume: 9 Issue: 1 Year: 2013 Page: 91-99
Author(s): Ravindra G. Kulkarnia, Stefan A. Laufer, Chandrashekhar V. M, Achaiah Garlapati

Cross-linked Mucoadhesive Microspheres based on Anionic Heteropolysaccharide for Nasal Delivery of Felodipine: Optimization and in vitro Evaluation

Journal: Drug Delivery Letters
Volume: 3 Issue: 2 Year: 2013 Page: 136-148
Author(s): Shobhita Mishra, Niraj Singh Patel, Manish Kumar, Kamla Pathak

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