Search Result "druggability"


Research Article

Possible Binding Mode Analysis of Pyrazolo-triazole Hybrids as Potential Anticancer Agents through Validated Molecular Docking and 3D-QSAR Modeling Approaches

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 5 Year: 2017 Page: 515-527
Author(s): Siekh Abdul Amin,Nilanjan Adhikari,Ram K. Agrawal,Tarun Jha,Shovanlal Gayen

Review Article

Calculating Water Thermodynamics in the Binding Site of Proteins – Applications of WaterMap to Drug Discovery

Journal: Current Topics in Medicinal Chemistry
Volume: 17 Issue: 23 Year: 2017 Page: 2586-2598
Author(s): Daniel Cappel,Woody Sherman,Thijs Beuming

Review Article

CRISPR-Cas in Medicinal Chemistry: Applications and Regulatory Concerns

Journal: Current Topics in Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2017 Page: 3308-3315
Author(s): Aliuska Duardo-Sanchez

Review Article

Alzheimer’s Drug Discovery Maze: A Snap View of the Past Decade’s Diverse Pharmacological Targets for the Disorder

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2017 Page: 305-318
Author(s): Donald Sikazwe,Raghunandan Yendapally,Sushma Ramsinghani,Malik Khan

Review Article

Targeting Apelinergic System in Cardiometabolic Disease

Journal: Current Drug Targets
Volume: 18 Issue: 15 Year: 2017 Page: 1785-1791
Author(s): Rui Guo,Olivia Rogers,Sreejayan Nair

Review Article

The Metabolomic Strategy in Tuberculosis Therapy

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 20 Issue: 3 Year: 2017 Page: 235-246
Author(s): Nitendra Kumar,Ashwinee Kumar Shreshtha,Sanjukta Patra

Research Article

Apicoplast Import Protein Tic20 A Promising Therapeutic Molecular Target for Plasmodium falciparum: An In Silico Approach for Therapeutic Intervention

Journal: Infectious Disorders - Drug Targets
Volume: 17 Issue: 3 Year: 2017 Page: 199-222
Author(s): Ravi C P. K. Srimath-Tirumala-Peddinti,Sandeep S. Kusuma,Deepthi Nammi,Nageswara R.R. Neelapu

Review Article

Nanotechnological Strategies to Improve Water Solubility of Commercially Available Drugs

Journal: Current Nanomedicine
Volume: 7 Issue: 2 Year: 2017 Page: 84-110
Author(s): Desiree Nedra Karunaratne,Isuru R. Ariyarathna,Dhanushi Welideniya,Asitha Siriwardhana,Dinara Gunasekera,Veranja Karunaratne

Review Article

CRISPR/Cas9 Editing to Facilitate and Expand Drug Discovery

Journal: Current Gene Therapy
Volume: 17 Issue: 4 Year: 2017 Page: 275-285
Author(s): Francis Robert,Sidong Huang,Jerry Pelletier

Research Article

Spices Chemoconstituents as Persuasive Inhibitor of S. typhimurium Virulent Protein L-asparaginase

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 1 Year: 2017 Page: 1433-1454
Author(s): Archana Vimal , Awanish Kumar

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