Search Result "druggability"


Review Article

The Potential of PI3K/AKT/mTOR Signaling as a Druggable Target for Endometrial and Ovarian Carcinomas

Journal: Current Drug Targets
Volume: 21 Issue: 1 Year: 2020 Page: 946-961
Author(s): Csongor György Lengyel,Sara Cecilia Altuna,Baker Shalal Habeeb,Dario Trapani,Shah Zeb Khan

Research Article

In Silico Drug Target Discovery Through Proteome Mining from M. tuberculosis: An Insight into Antivirulent Therapy

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 23 Issue: 3 Year: 2020 Page: 253-268
Author(s): Shreya Bhattacharya,Puja Ghosh,Debasmita Banerjee,Arundhati Banerjee,Sujay Ray

Review Article

p53: An Attractive Therapeutic Target for Cancer

Journal: Current Medicinal Chemistry
Volume: 27 Issue: 2 Year: 2020 Page: 3706-3734
Author(s): Krupa R. Patel,Hitesh D. Patel

Review Article

Emergence and Reemergence of Human Coronaviruses: Spike Protein as the Potential Molecular Switch and Pharmaceutical Target

Journal: Current Pharmaceutical Design
Volume: 26 Issue: 0 Year: 2020 Page: 1-14
Author(s): Fahim Ahmad,Mohammad A. Kamal,Babu L. Tekwani

Review Article

Clinical Relevance of Alternative Lengthening of Telomeres in Cancer

Journal: Current Topics in Medicinal Chemistry
Volume: 20 Issue: 6 Year: 2020 Page: 485-497
Author(s): Guilherme G. da Silva,Karollyne S. Morais,Daniel S. Arcanjo,Diêgo M. de Oliveira

Review Article

Adult Neurogenesis in Epileptogenesis: An Update for Preclinical Finding and Potential Clinical Translation

Journal: Current Neuropharmacology
Volume: 18 Issue: 6 Year: 2020 Page: 464-484
Author(s): Liying Chen,Yi Wang,Zhong Chen

Research Article

Design, Synthesis, Docking and Computational Pharmacokinetic Profiling of New Pyrazolinyl Thiazolinone Biheterocycles as Potent Antimicrobial Agents

Journal: Letters in Drug Design & Discovery
Volume: 17 Issue: 1 Year: 2020 Page: 1342-1354
Author(s): Vinutha V. Salian,Badiadka Narayana,Balladka K. Sarojini,Sharath Chandra K.,Anupam G. Lobo

Subtractive Genomics Approaches: Towards Anti- Bacterial Drug Discovery

Ebook: Vascularization in Tissue Engineering

Volume: 8 Year: 2020
Author(s): Fatima Shahid,Muhammad Shehroz,Tahreem Zaheer,Amjad Ali
Doi: 10.2174/97898114123871190801
Research Article

Kaempferol as a Potential PAK4 Inhibitor in Triple Negative Breast Cancer: Extra Precision Glide Docking and Free Energy Calculation

Journal: Current Drug Discovery Technologies
Volume: 17 Issue: 5 Year: 2020 Page: 682-695
Author(s): Michael A. Arowosegbe,Oluwamuyiwa T. Amusan,Segun A. Adeola,Oluwatosin B. Adu,Israel A. Akinola,Bimpe F. Ogungbe,Olaposi I. Omotuyi,Gbemisola M. Saibu,Adewale J. Ogunleye,Ramon I. Kanmodi,Nekabari E. Lugbe,Oluwafemi J. Ogunmola,Damilola C. Ajayi,Sedoten O. Ogun,Faith O. Oyende,Ahmed O. Bello,Peter G. Ishola,Patrick E. Obasieke

Review Article

From Recognition to Reaction Mechanism: An Overview on the Interactions between HIV-1 Protease and its Natural Targets

Journal: Current Medicinal Chemistry
Volume: 27 Issue: 1 Year: 2020 Page: 2514-2549
Author(s): Monsurat M. Lawal,Zainab K. Sanusi,Thavendran Govender,Glenn E.M. Maguire,Bahareh Honarparvar,Hendrik G. Kruger

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