Search Result "hERG"


Implications of Dynamic Occupancy, Binding Kinetics, and Channel Gating Kinetics for hERG Blocker Safety Assessment and Mitigation

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 16 Year: 2016 Page: 1792-1818
Author(s): Robert A. Pearlstein,K. Andrew MacCannell,Gül Erdemli,Sarita Yeola,Gabriel Helmlinger,Qi-Ying Hu,Ramy Farid,William Egan,Steven Whitebread,Clayton Springer,Jeremy Beck,Hao-Ran Wang,Mateusz Maciejewski,Laszlo Urban,José S. Duca

Artificial Neural Network Analysis of Pharmacokinetic and Toxicity Properties of Lead Molecules for Dengue Fever, Tuberculosis and Malaria

Journal: Current Computer-Aided Drug Design
Volume: 12 Issue: 1 Year: 2016 Page: 52-61
Author(s): Shahul H. Nilar,Suresh B. Lakshminarayana,Ngai Ling Ma,Thomas H. Keller,Francesca Blasco,Paul W. Smith

Drug-induced Inhibition and Trafficking Disruption of ion Channels: Pathogenesis of QT Abnormalities and Drug-induced Fatal Arrhythmias

Journal: Current Cardiology Reviews
Volume: 12 Issue: 2 Year: 2016 Page: 141-154
Author(s): Luigi X. Cubeddu

The Impact of Opioids on Cardiac Electrophysiology

Journal: Current Cardiology Reviews
Volume: 12 Issue: 1 Year: 2016 Page: 27-36
Author(s): Erich F. Wedam,Mark C. Haigney

Immunophilins: Structures, Mechanisms and Ligands

Journal: Current Molecular Pharmacology
Volume: 9 Issue: 1 Year: 2016 Page: 37-47
Author(s): Amaravadhi Harikishore,Ho Sup Yoon

Computer-Aided Drug Discovery and Design Targeting Ion Channels

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 16 Year: 2016 Page: 1819-1829
Author(s): Qiansen Zhang,Zhaobing Gao,Huaiyu Yang

The Recent Development of α7 Nicotinic Acetylcholine Receptor (nAChR) Ligands as Therapeutic Candidates for the Treatment of Central Nervous System (CNS) Diseases

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 14 Year: 2016 Page: 2134-2151
Author(s): Corinne Beinat,Samuel D. Banister,Marco Herrera,Michael Kassiou

Natural Products based P-glycoprotein Activators for Improved β-amyloid Clearance in Alzheimer’s Disease: An in silico Approach

Journal: Central Nervous System Agents in Medicinal Chemistry
Volume: 16 Issue: 1 Year: 2016 Page: 50-59
Author(s): Pravin Shinde,Nikhil Vidyasagar,Sivakami Dhulap,Abhijeet Dhulap,Raj Hirwani

Research Article

Tramadol Induced QTc-Interval Prolongation: Prevalence, Clinical Factors and Correlation to Plasma Concentrations

Journal: Current Drug Safety
Volume: 11 Issue: 3 Year: 2016 Page: 206-214
Author(s):

Relationship Between Carbapenems Structure and Minimal Inhibitory Concentration Selected Bacterial Strains

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 5 Year: 2016 Page: 422-428
Author(s): Monika Marczak,Tomasz Grabowski

Previous   Next

Go To   Results 1 - 1 of 44

Filter Result

Volume Year
Content Type
Ads
© 2024 Bentham Science Publishers | Privacy Policy