Search Result "imatinib"


Research Article

Design, Synthesis and Biological Evaluation of Betulinic Acid Derivatives as New Antitumor Agents for Leukemia

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 1 Year: 2017 Page: 1777-1785
Author(s): Fernanda Waechter,Gloria N.S. da Silva,Julia B. Willig,Cristiane B. de Oliveira,Bruna D. Vieira,Daniela B.B. Trivella,Aline R. Zimmer,Andreia Buffon,Diogo A. Pilger,Simone C.B. Gnoatto

Review Article

Insight to Pharmacokinetics of TKIs: Optimizing Practical Guidelines for Individualized Therapy

Journal: Current Drug Metabolism
Volume: 18 Issue: 3 Year: 2017 Page: 199-206
Author(s): Ruiqing Wang,Chaoqin Zhong,Chen Zhang,Mingqiang Hua,Daoxin Ma

Review Article

Cellular and Molecular Networks in Chronic Myeloid Leukemia: The Leukemic Stem, Progenitor and Stromal Cell Interplay

Journal: Current Drug Targets
Volume: 18 Issue: 4 Year: 2017 Page: 377-388
Author(s): Danilo Perrotti,Giovannino Silvestri,Lorenzo Stramucci,Justine Yu,Rossana Trotta

Review Article

Heterocyclic Analogues as Kinase Inhibitors: A Focus Review

Journal: Current Topics in Medicinal Chemistry
Volume: 17 Issue: 22 Year: 2017 Page: 2482-2494
Author(s): Vikas Sharma,Raj Kamal,Vipin Kumar

Review Article

Development of a Predictive Pharmacophore Model and a 3D-QSAR Study for an in silico Screening of New Potent Bcr-Abl Kinase Inhibitors

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2017 Page: 188-204
Author(s): Eleni Vrontaki,Georgia Melagraki,Stella Voskou,Marios S. Phylactides,Thomas Mavromoustakos,Marina Kleanthous,Antreas Afantitis

Review Article

The Polyhedric Abl Kinases and their Pharmacologic Inhibitors

Journal: Current Enzyme Inhibition
Volume: 13 Issue: 2 Year: 2017 Page: 129-138
Author(s): Elisa Lupino, Marco Piccinini

Review Article

Repurposing Pharmaceuticals as Neuroprotective Agents for Cerebral Malaria

Journal: Current Clinical Pharmacology
Volume: 12 Issue: 2 Year: 2017 Page: 62-72
Author(s): Hannah M. Brooks,Michael T. Hawkes

Review Article

Small-Cell Lung Cancer: Clinical Management and Unmet Needs New Perspectives for an Old Problem

Journal: Current Drug Targets
Volume: 18 Issue: 3 Year: 2017 Page: 341-362
Author(s): Giuseppe Lo Russo,Marianna Macerelli,Marco Platania,Nicoletta Zilembo,Milena Vitali,Diego Signorelli,Claudia Proto,Monica Ganzinelli,Rosaria Gallucci,Francesco Agustoni,Gianpiero Fasola,Filippo de Braud,Marina Chiara Garassino

Review Article

Recurrent Fusion Genes in Leukemia: An Attractive Target for Diagnosis and Treatment

Journal: Current Genomics
Volume: 18 Issue: 5 Year: 2017 Page: 378-384
Author(s): Yuhui Wang,Nan Wu,Duo Liu,Yan Jin

Research Article

Apoptotic Effects of Some Tetrahydronaphthalene Derivatives on K562 Human Chronic Myelogenous Leukemia Cell Line

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 1 Year: 2017 Page: 1924-1930
Author(s): Asli Koc,Tulin Ozkan,Yalda Hekmatshoar,A. Selen Gurkan-Alp,Fugen Aktan,Zeliha Buyukbingol,Asuman Sunguroglu,Erdem Buyukbingol,Arzu Zeynep Karabay

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