Search Result "thiourea"


Research Article

Synthesis, Structural Studies and Biological Evaluation of Halogen Derivatives of 1,3-Disubstituted Thiourea

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 6 Year: 2017 Page: 636-646
Author(s): Anna Bielenica, Karolina Stepien, Aleksandra Sawczenko, Tadeusz Lis, Anna E. Koziol, Silvia Madeddu, David Collu, Filippo Iuliano, Anita Kosmider, Marta Struga

Research Article

Novel Thiourea Derivatives Bearing Sulfonamide Moiety as Anticancer Agents Through COX-2 Inhibition

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 10 Year: 2017 Page: 1411-1425
Author(s): Mostafa M. Ghorab,Mohamed S.A. El-Gaby,Mansour S. Alsaid,Yaseen A.M.M. Elshaier,Aiten M. Soliman,Fardous F. El-Senduny,Farid A. Badria,Abdelrahman Y.A. Sherif

Research Article

Solvent-Free Synthesis of Thiobarbituric Acids Using Amberlyst-15 as a Green Catalyst

Journal: Current Green Chemistry
Volume: 4 Issue: 1 Year: 2017 Page: 50-56
Author(s): Manish M. Katiya,Madhukar G. Dhonde,Jayant M. Gajbhiye

Research Article

Microwave Assisted Extraction and in vitro Evaluation of urease Inhibition Potential of Stem Bark of Terminalia arjuna

Journal: Current Microwave Chemistry
Volume: 4 Issue: 3 Year: 2017 Page: 199-204
Author(s): Sarita Khatkar,Arun Nanda,S.H. Ansari

Research Article

β-Cyclodextrin (β-CD) as a Supramolecular Catalyst for the Synthesis of Isoxazoles and Thiopyrimidines and their Antimicrobial Screening

Journal: Letters in Organic Chemistry
Volume: 14 Issue: 2 Year: 2017 Page: 93-102
Author(s): Asha V. Chate,Charansingh H. Gill

Research Article

6-Benzothiazolyl Ureas, Thioureas and Guanidines are Potent Inhibitors of ABAD/17β-HSD10 and Potential Drugs for Alzheimer"s Disease Treatment: Design, Synthesis and in vitro Evaluation

Journal: Medicinal Chemistry
Volume: 13 Issue: 4 Year: 2017 Page: 345-358
Author(s): Ondrej Benek, Lukas Hroch, Laura Aitken, Rafael Dolezal, Patrick Guest, Marketa Benkova, Ondrej Soukup, Karel Musil, Kamil Kuca, Terry K. Smith, Frank Gunn-Moore, Kamil Musilek

Research Article

Synthesis of N-glycosylated Dihydropyrimidones – A Novel Approach Using Epoxy Sugar

Journal: Letters in Organic Chemistry
Volume: 14 Issue: 3 Year: 2017 Page: 192-197
Author(s): K. R. Subimol,S. Arul Antony

Research Article

Bisthiourea Derivatives of Dipeptide Conjugated Benzo[d]isoxazole as a New Class of Therapeutics: Synthesis and Molecular Docking Studies

Journal: Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2017 Page: 123-133
Author(s): Honnegowdanahally K. Kumara,Doddahindaiah M. Suyoga Vardhan,J. Shiva Kumar,D. Channe Gowda

Research Article

4-Methylumbelliferones Analogues as Anticancer Agents: Synthesis and in Cell Pharmacological Studies

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 4 Year: 2017 Page: 576-589
Author(s): Ri-Zhen Huang,Shi-Xian Hua,Cai-Yi Wang,Ying-Ming Pan,Jian-Mei Qin,Zhan-Yu Ding,Ye Zhang,Heng-Shan Wang

Research Article

Quorum Sensing Inhibitor Activities of Celecoxib Derivatives in Pseudomonas aeruginosa

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 5 Year: 2017 Page: 613-618
Author(s): Seyhan Ulusoy,Sevil Senkardes,Inci Coskun,Gulgun Bosgelmez-Tınaz,Laurent Soulere,Yves Queneau,S. Guniz Kucukguzel

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