Search Result "tyrosine kinase inhibitor"


Review Article

Recent Patents on the Development of c-Met Kinase Inhibitors

Journal: Recent Patents on Anti-Cancer Drug Discovery
Volume: 15 Issue: 3 Year: 2020 Page: 228-238
Author(s): Xiangming Xu,Lei Yao

Review Article

Targeting Small Molecule Tyrosine Kinases by Polyphenols: New Move Towards Anti-tumor Drug Discovery

Journal: Current Drug Discovery Technologies
Volume: 17 Issue: 5 Year: 2020 Page: 585-615
Author(s): Nikhil S. Sakle,Shweta A. More,Sachin A. Dhawale,Santosh N. Mokale

Review Article

Computational Approaches for the Design of (Mutant-)Selective Tyrosine Kinase Inhibitors: State-of-the-Art and Future Prospects

Journal: Current Topics in Medicinal Chemistry
Volume: 20 Issue: 1 Year: 2020 Page: 1522-1533
Author(s): Prashant S. Kharkar

Review Article

Studies on Structures and Functions of Kinases leading to Prostate Cancer and Their Inhibitors

Journal: Current Enzyme Inhibition
Volume: 16 Issue: 1 Year: 2020 Page: 90-105
Author(s): Anantha Naik Nagappa,Shvetank Bhatt,Jovita Kanoujia

Mini-Review Article

Inhibitor Binding Sites in the Protein Tyrosine Phosphatase SHP-2

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 20 Issue: 1 Year: 2020 Page: 1017-1030
Author(s): Haonan Zhang,Zhengquan Gao,Chunxiao Meng,Xiangqian Li,Dayong Shi

Bruton’s Tyrosine Kinase Signaling and Advancement in Multiple Myeloma Therapy

Ebook: Vascularization in Tissue Engineering

Volume: 1 Year: 2020
Author(s): Krishne Gowda,Max Von Suskil,Omar Al-Adat,Jennifer Dang,Kuntal Bhowmick,Prachi S. Narayan,Shantu G Amin,Manoj K. Pandey
Doi: 10.2174/97898114581181200101
Review Article

Carbazole Derivatives as Kinase-Targeting Inhibitors for Cancer Treatment

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 20 Issue: 6 Year: 2020 Page: 444-465
Author(s): Jessica Ceramella,Domenico Iacopetta,Alexia Barbarossa,Anna Caruso,Fedora Grande,Maria Grazia Bonomo,Annaluisa Mariconda,Pasquale Longo,Saturnino Carmela,Maria Stefania Sinicropi Stefania Sinicropi

Review Article

Therapeutic Journey of Pyrazolines as EGFR Tyrosine Kinase Inhibitors: An Insight into Structure-Activity Relationship

Journal: Current Bioactive Compounds
Volume: 16 Issue: 9 Year: 2020 Page: 1260-1272
Author(s): Navdeep Singh,Monika Gupta

Letter to the Editor

Lapatinib as a Dual Tyrosine Kinase Inhibitor Unexpectedly Activates Akt in MDA-MB-231 Triple-Negative Breast Cancer Cells

Journal: Letters in Drug Design & Discovery
Volume: 17 Issue: 8 Year: 2020 Page: 1060-1063
Author(s): Parham Jabbarzadeh Kaboli,King-Hwa Ling

Research Article

Heterocyclization of 2-(2-phenylhydrazono)cyclohexane-1,3-dione to Synthesis Thiophene, Pyrazole and 1,2,4-triazine Derivatives with Anti-Tumor and Tyrosine Kinase Inhibitions

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 20 Issue: 1 Year: 2020 Page: 1209-1220
Author(s): Rafat M. Mohareb,Ensaf S. Alwan

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