Search Result "tyrosine kinase inhibitors"


Review Article

Tyrosine Kinase Inhibitors (TKIs) in Lung Cancer Treatment: A Comprehensive Analysis

Journal: Current Cancer Drug Targets
Volume: 21 Issue: 1 Year: 2021 Page: 55-69
Author(s): Sivakumar Murugesan,Jayakumar Murugesan,Seedevi Palaniappan,Sivasankar Palaniappan,Tamilselvi Murugan,Shahid S. Siddiqui,Sivakumar Loganathan

Mini-Review Article

Computational and Biological Investigations on Abl1 Tyrosine Kinase: A Review

Journal: Current Drug Targets
Volume: 22 Issue: 1 Year: 2021 Page: 38-51
Author(s): Masilamani Elizabeth Sobhia,G. Siva Kumar,Antara Mallick,Harmanpreet Singh,Kranthi Kumar,Meenakshi Chaurasiya,Narendra Gera,Sindhuja Deverakonda,Vinay Baghel

Review Article

Pharmacologic Evidence of Green Tea in Targeting Tyrosine Kinases

Journal: Current Reviews in Clinical and Experimental Pharmacology
Volume: 16 Issue: 3 Year: 2021 Page: 239-246
Author(s): Joyce T.S. Li,Kam L. Hon,Alexander K.C. Leung,Vivian W.Y. Lee

Case Report

Concomitant use of Tyrosine-Kinase Inhibitor and Mepolizumab in AsthmaSecondary to Chronic Myeloid Leukemia with Hypereosinophilia

Journal: Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry
Volume: 20 Issue: 4 Year: 2021 Page: 389-393
Author(s): Antonio Gidaro,Emanuele Salvi,Maria Cristina Carraro,Roberta Simona Rossi,Roberto Castelli

Research Article

In vitro Measurement and In vivo Prediction of Time-Dependent Inhibitory Effects of Three Tyrosine Kinase Inhibitors on CYP3A Activity

Journal: Current Drug Metabolism
Volume: 22 Issue: 1 Year: 2021 Page: 802-810
Author(s): Liyan Wang,Tingting Zhao,Yunxiang Wang,Banglian Hu,Jianfei Tao,Jinshan Ke,Tingfei Wei,Guangbo Ge,Qiang Meng,Changyuan Wang,Qi Liu,Huijun Sun,Jingjing Wu,Yanwei Chen

Research Article

New Approaches for the Synthesis of Heterocyclic Compounds Corporating Benzo[d]imidazole as Anticancer Agents, Tyrosine, Pim-1 Kinases Inhibitions and their PAINS Evaluations

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 21 Issue: 3 Year: 2021 Page: 279-294
Author(s): Rafat M. Mohareb,Yara R. Milad,Bahaa M. Mostafa,Reem A. El-Ansary

Review Article

Recent Advances of Small Molecule Focal Adhesion Kinase (FAK) Inhibitors as Promising Anticancer Therapeutics

Journal: Current Medicinal Chemistry
Volume: 28 Issue: 0 Year: 2021 Page: 1-13
Author(s): Pengcheng Lv,Kun Chen,Hai-Liang Zhu

Research Article

Design, Synthesis, Molecular Docking, and Anticancer Evaluation of Pyrazole Linked Pyrazoline Derivatives with Carbothioamide Tail as EGFR Kinase Inhibitors

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 21 Issue: 1 Year: 2021 Page: 42-60
Author(s): Farah Nawaz,Ozair Alam,Ahmad Perwez,Moshahid A. Rizvi,Mohd. Javed Naim,Nadeem Siddiqui,Jannat ul Firdaus,Shakilur Rahman,Mukund Jha,Aadil A. Sheikh

Research Article

Fragment-Based Drug Design of Antitumoral Molecules Polo-like kinase 1 inhibitors: in-silico approach

Journal: Letters in Drug Design & Discovery
Volume: 18 Issue: 0 Year: 2021 Page: 1-18
Author(s): Yacine Benguerba,Nour El Houda Hammoudi,Widad Sobhi,Ayoub Attoui

Research Article

A New Series of Antileukemic Agents: Design, Synthesis, In Vitro and In Silico Evaluation of Thiazole-Based ABL1 Kinase Inhibitors

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 21 Issue: 9 Year: 2021 Page: 1099-1109
Author(s): Ebru Zeytün,Mehlika D. Altıntop,Belgin Sever,Ahmet Özdemir,Doha E. Ellakwa,Zeynep Ocak,Halil I. Ciftci,Masami Otsuka,Mikako Fujita,Mohamed O. Radwan

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